Isoetharine mesylate salt

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断

Isoetharine Mesylate Salt 是一种 β-肾上腺素能受体激动剂。它也是孕烷 X 受体 (PXR) 激活剂，能够上调 CYP450 表达。

Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.(In Vitro):Isoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.(In Vivo):Isoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.

Isoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.

Isoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.

Isoetarine mesilate

Angiogenesis

Adrenergic Receptor

β-adrenergic receptor| PXR

Others

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7279-75-6

335.42

C14H25NO6S

>98% (HPLC)

DMSO:199.7 mM;Water:199.7 mM

CS(O)(=O)=O.CCC(NC(C)C)C(O)c1ccc(O)c(O)c1

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(-20℃)

With Ice Pack

≥ 2 years